Treeline Biosciences

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Treeline Biosciences, Inc.

22 Investors
Biotechnology & Drug Discovery
WATERTOWN, MA

Treeline Biosciences is a clinical-stage biotechnology company developing precision medicines for cancer and other serious diseases. Founded in 2021 with significant financial backing, the company focuses on historically difficult-to-drug molecular targets in oncology and has recently advanced three distinct therapeutic candidates into Phase 1 clinical trials.

Products & Team

TLN-372 (KRAS Inhibitor)

Oncology TherapeuticSeed

TLN-372 is an internally developed small molecule inhibitor designed to target multiple mutations in the KRAS gene. These mutations are common drivers in various solid tumors, including those affecting the lung, colon, and pancreas.

Value Proposition

This therapeutic addresses the long-standing challenge of effectively drugging the KRAS protein, which is one of the most frequently mutated oncogenes in human cancers and has been notoriously difficult to inhibit.

Pain Points

The company addresses the critical need for effective treatments for patients with cancers that have either become resistant to existing therapies or have historically lacked targeted treatment options due to the complexity of their underlying genetic drivers.

Small molecule inhibitorDesigned to broadly target multiple KRAS mutationsDeveloped for solid tumors such as lung, colon, and pancreas cancer

Joshua H. Bilenker, M.D.

Company Signatory
Chief Executive Officerat Treeline Biosciences, Inc.
Joined Treeline Biosciences, Inc.
September 2025

Ali Satvat

Directorat Treeline Biosciences, Inc.
Joined Treeline Biosciences, Inc.
September 2025
Industry
Biotechnology
Primary business sector
Founded
2025
Year established
Location
WATERTOWN, MA
Primary headquarters

Funding History

Total Raised:
$200.1M
E

Equity, Option to Acquire Offering

August 2025
$250.0M
Target
Progress
80%
Raised
$200.1M
Target
$250.0M
#000185661925000002

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